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Signaling Pathways - Glutamate (Metabotropic) Group I Receptors - Histamine H1 Receptors

15件产品中的 1-10

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  1. NPS 2390
    B5532 NPS 2390
    Target: Glutamate (Metabotropic) Group I Receptors
    Summary: I型mGlu拮抗剂
      Soluble in DMSO
  2. CHPG
    B6569 CHPG
    Target: Glutamate (Metabotropic) Group I Receptors
    Summary: mGlu5代谢型谷氨酸受体激动剂
  3. 2-Pyridylethylamine dihydrochloride
    B7072 2-Pyridylethylamine dihydrochloride
    Target: Histamine H1 Receptors
    Summary: 组胺H1受体激动剂
      <9.75 mg/mL
      <19.51 mg/mL
  4. Azelastine HCl
    B1568 Azelastine HCl
    中文名: 盐酸氮卓斯汀
    Target: Histamine H1 Receptors
    Summary: 有效的,第二代,选择性的组胺受体拮抗剂
      ≥20.92 mg/mL
      ≥5.42 mg/mL
  5. Rupatadine Fumarate
    B1566 Rupatadine Fumarate
     1 Citation
    中文名: 富马酸卢帕他定
    Target: Histamine H1 Receptors|PAFR
    Summary: PAF和组胺(H1)受体的抑制剂
      ≥11.75 mg/mL
      insoluble in H2O
  6. Pemirolast potassium
    B1563 Pemirolast potassium
    中文名: 吡嘧司特钾
    Target: Histamine H1 Receptors
    Summary: 组胺H1受体拮抗剂
      ≥5.37 mg/mL
      ≥85.4 mg/mL
  7. Hydroxyzine 2HCl
    B1549 Hydroxyzine 2HCl
    中文名: 羟嗪二盐酸盐
    Target: Histamine H1 Receptors
    Summary: 组胺H1受体拮抗剂
      ≥21.5 mg/mL
      ≥9.5 mg/mL
  8. Cyclizine 2HCl
    B1548 Cyclizine 2HCl
    中文名: 氧杂蒽酮
    Target: Histamine H1 Receptors
    Summary: 组胺H1受体拮抗剂
      Soluble in DMSO
  9. Cetirizine DiHCl
    B1547 Cetirizine DiHCl
    中文名: 盐酸西替利嗪
    Target: Histamine H1 Receptors
    Summary: H1受体反向激动剂
      ≥23.09 mg/mL
      ≥2.66 mg/mL
  10. Terfenadine
    A8534 Terfenadine
    中文名: 特非那定
    Target: Voltage-gated Potassium (KV) Channels|Histamine H1 Receptors|Inward Rectifier Potassium (Kir) Channels
    Summary: 组胺H1受体拮抗剂
      ≥18 mg/mL
      insoluble in H2O

15件产品中的 1-10

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