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- N2133 7-Ethyl-10-hydroxycamptothecinTarget: TopoisomerasesSummary: TOPO I抑制剂
- B4745 (S)-10-Hydroxycamptothecin中文名: 羟喜树碱Target: TopoisomerasesSummary: 拓扑异构酶I抑制剂
- B1801 Norfloxacin中文名: 诺氟沙星Target: TopoisomerasesSummary: 拓扑异构酶抑制剂
- A4536 Fostriecin sodium saltTarget: PP1|PP2A|Topoisomerases|PP4Summary: 抗肿瘤抗生素
- A1832 Doxorubicin (Adriamycin) HCl2 Citation中文名: 盐酸多柔比星,盐酸阿霉素Target: TopoisomerasesSummary: 抗肿瘤抗生素,抑制TOPO II。
- B5082 FR 139317Target: endothelin receptorSummary: 选择性ETA内皮素受体拮抗剂
- B6431 Zinc protoporphyrin IX2 Citation中文名: 锌原卟啉Target: Guanylyl Cyclases|Heme oxygenaseSummary: 血红素加氧酶抑制剂
- B7382 Ellipticine中文名: 玫瑰树碱,椭圆玫瑰树碱Target: TopoisomerasesSummary: DNA拓扑异构酶II抑制剂
- B7641 YC 1中文名: 利非西呱Target: Guanylyl CyclasesSummary: 可溶性鸟苷酸环化酶(sGC)激活剂