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- A8621 Bestatin hydrochloride中文名: 盐酸乌苯美司Target: AminopeptidasesSummary: 氨肽酶N(APN/CD13)和氨肽酶B抑制剂。
- B2224 Etravirine (TMC125)中文名: 依曲韦林Target: Reverse TranscriptasesSummary: 逆转录酶抑制剂
- B1946 Foscarnet Sodium中文名: 膦甲酸钠Target: Reverse Transcriptases|RNA PolymerasesSummary: 逆转录酶抑制剂
- A4364 Methazolamide中文名: 醋甲唑胺Target: Carbonic AnhydrasesSummary: 碳酸酐酶抑制剂
- A1755 Tenofovir Disoproxil Fumarate中文名: 富马酸替诺福韦酯Target: Reverse TranscriptasesSummary: 抗逆转录制剂(HIV-1 RT 抑制剂)
- A5354 Zonisamide中文名: 唑尼沙胺Target: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Carbonic Anhydrases|Calcium-Activated Potassium (KCa) ChannelsSummary: 抗惊厥和机械效应的抗癫痫药
- A8410 Didanosine中文名: 去羟肌苷Target: Reverse TranscriptasesSummary: 逆转录酶抑制剂
- A8397 Chlorothiazide中文名: 氯噻嗪Target: Carbonic AnhydrasesSummary: 碳酸酐酶抑制剂
- A2197 Dacarbazine中文名: 达卡巴嗪Target: DNA AlkylatingSummary: 抗肿瘤(恶性黑色素瘤和肉瘤)
- A3237 Betulinic acid中文名: 白桦脂酸,桦木酸Target: Aminopeptidases|Topoisomerases|HIVSummary: 抗HIV和抗肿瘤化合物,五环三萜类化合物