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- A4447 2,3-DCPE hydrochlorideTarget: Apoptosis InducersSummary: Bcl-XL蛋白表达下调剂
- B1874 4μ8C2 CitationTarget: Inositol-requiring enzyme 1 (IRE1)Summary: IRE1 Rnase抑制剂
- A3021 GDC-0449 (Vismodegib)1 Citation中文名: 维莫德吉Target: P-glycoprotein (P-gp)|HedgehogSummary: Hedgehog拮抗剂
- A3956 ZosuquidarTarget: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)Summary: MDR调节剂
- A4390 Pemetrexed1 Citation中文名: 培美曲塞二钠盐Target: Thymidylate Synthase|DHFR|GARFTSummary: TS、DHFR、GARFT和AICARFT抑制剂