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- A1036 Thrombin Receptor Activator for Peptide 5 (TRAP-5)Target: Thrombin ReceptorSummary: Thrombin Receptor Activator for Peptide 5
- A3185 AR-C155858Target: Monocarboxylate transporters (MCTs)Summary: MCT1和MCT2抑制剂
- B1111 N6022Target: S-nitrosoglutathione reductaseSummary: GSNOR抑制剂
- A4024 Danoprevir (RG7227)中文名: 丹诺瑞韦Target: HCV ProteasesSummary: HCV NS3/4A蛋白酶抑制剂