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- B2219 EHop-0161 CitationTarget: RacSummary: Rac1/Rac3 GTPase抑制剂
- B3209 TriapineTarget: Ribonucleotide ReductasesSummary: 核糖核苷酸还原酶(ribonucleotide reductase)抑制剂
- A4430 Sivelestat sodium salt中文名: 西维来司钠Target: ElastasesSummary: 白细胞弹性蛋白酶抑制剂
- A8809 Vorapaxar中文名: 沃拉帕沙Target: Protease-Activated ReceptorsSummary: PAR-1拮抗剂