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- A3374 Dronedarone中文名: 决奈达隆Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channelSummary: CYP3A4和2D6抑制剂
- A1932 (-)-Huperzine A中文名: 石杉碱甲Target: NMDA Receptors|AChESummary: NMDA受体拮抗剂/AChE抑制剂
- A4130 ENMD-2076Target: Aurora Kinases|FLT3|RET|Src|VEGFR3/FLT4|NTRK1/TRKA|CSF-1R/c-FmsSummary: Aurora A/Flt3的选择性抑制剂
- A3237 Betulinic acid中文名: 白桦脂酸,桦木酸Target: Aminopeptidases|Topoisomerases|HIVSummary: 抗HIV和抗肿瘤化合物,五环三萜类化合物