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- A3003 MDV3100 (Enzalutamide)12 Citation中文名: 恩杂鲁胺Target: Androgen ReceptorsSummary: 雄激素受体拮抗剂。
- A2150 AndarineTarget: Androgen ReceptorsSummary: 雄激素受体拮抗剂
- A4492 NU 9056Target: Histone Acetyltransferases (HATs)Summary: KAT5(Tip60)HAT抑制剂
- A4488 Anacardic acid中文名: 漆树酸Target: Histone Acetyltransferases (HATs)Summary: HAT抑制剂
- B1182 ABC294640中文名: 奥帕尼布Target: SKSummary: 鞘氨醇激酶2抑制剂