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- A8641 LEE011中文名: 瑞博西利,瑞博西林Target: Cyclin-Dependent KinasesSummary: CDK4/6抑制剂
- A3541 LCL1611 CitationTarget: Inhibitor of apoptosis proteins (IAP)Summary: IAPs拮抗剂
- A4135 Tofacitinib (CP-690550) Citrate2 Citation中文名: 托法替尼Target: JAKSummary: JAK抑制剂
- A4317 Apremilast (CC-10004)中文名: 阿普斯特Target: Phosphodiesterases (PDEs)Summary: PDE4抑制剂