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- A4326 TAK-700 (Orteronel)2 CitationTarget: human lyaseSummary: 人17,20-裂解酶抑制剂
- B4890 HPOB1 CitationTarget: Histone Deacetylases (HDACs)Summary: HDAC6抑制剂
- A4091 PCI-340511 CitationTarget: Histone Deacetylases (HDACs)Summary: HDAC8抑制剂
- A1882 Cediranib (AZD217)中文名: 西地尼布Target: VEGFRSummary: VEGFR受体高度有效的抑制剂