搜索结果: 'research-area epigenetics dna-methyltransferase'
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- A1913 RG 1083 CitationTarget: DNA MethyltransferasesSummary: DNA甲基转移酶抑制剂
- A1912 Lomeguatrib中文名: 罗米鲁曲Target: O6-methylguanine-DNA-methyl-transferase (MGMT)Summary: MGMT抑制剂
- A8315 NU7441 (KU-57788)4 CitationTarget: PI3K|DNA-PKSummary: DNA-PK抑制剂
- A8182 3-Deazaneplanocin A (DZNep) hydrochloride1 Citation中文名: 3-去氮腺嘌呤A盐酸盐Target: EZH2Summary: SAHH和EZH2抑制剂
- A4084 Vorinostat (SAHA, MK0683)9 Citation中文名: 伏立诺他Target: Histone Deacetylases (HDACs)Summary: HDAC抑制剂
- A1769 KU-00606481 CitationTarget: PI3K|DNA-PKSummary: DNA-PK/PI3-K双重抑制剂
- A3872 TH-302Summary: 低氧激活的前体药物,抑制H460/HT29细胞生长
- A4096 Belinostat (PXD101)2 Citation中文名: 贝利司他Target: Histone Deacetylases (HDACs)Summary: 羟肟酸型HDAC抑制剂
- A4111 VX-680 (MK-0457,Tozasertib)中文名: 陶扎色替Target: Aurora KinasesSummary: Aurora 激酶抑制剂
- B2290 Beta-Lapachone中文名: β-拉帕醌Target: TopoisomerasesSummary: 选择性DNA拓扑异构酶I抑制剂