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- A4447 2,3-DCPE hydrochlorideTarget: Apoptosis InducersSummary: Bcl-XL蛋白表达下调剂
- A2597 Brivanib (BMS-540215)中文名: 布立尼布Target: VEGFR|FGFR|Flk1Summary: VEGFR-2的ATP竞争性抑制剂
- B3709 Midostaurin (PKC412)中文名: 米哚妥林Target: PKC|PKA|KDR|Flk1|PPK|c-Syk|CDK1/CyclinBSummary: PKC抑制剂
- B5437 Decanoyl-RVKR-CMKTarget: Subtilisin/Kex2p-like proprotein convertaseSummary: 枯草杆菌蛋白酶/Kex2p样前蛋白转化酶抑制剂
- A3146 AGI-6780Target: IDH2Summary: IDH2/R140Q突变抑制剂