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- A8366 ARRY-380Target: HER2Summary: 酪氨酸激酶HER2和P95-HER2抑制剂。
- B7207 SecinH3Target: Guanine nucleotide exchange factors (GEFs)Summary: Sec7特异性GEF抑制剂
- A2097 Ifosfamide中文名: 异环磷酰胺Target: DNA AlkylatingSummary: 细胞抑制剂
- B4357 UNC2881Target: Mer tyrosine kinaseSummary: Mer酪氨酸激酶抑制剂
- A2197 Dacarbazine中文名: 达卡巴嗪Target: DNA AlkylatingSummary: 抗肿瘤(恶性黑色素瘤和肉瘤)
- A3145 Afatinib dimaleate中文名: 马来酸阿法替尼Target: EGFR|HER2Summary: EGFR抑制剂
- A8528 TAK-285Target: EGFR|HER2Summary: HER2/EGFR(HER1)抑制剂