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- A8366 ARRY-380Target: HER2Summary: 酪氨酸激酶HER2和P95-HER2抑制剂。
- B5750 ML 281Target: STKSummary: 丝氨酸/苏氨酸激酶STK33抑制剂
- A3021 GDC-0449 (Vismodegib)1 Citation中文名: 维莫德吉Target: P-glycoprotein (P-gp)|HedgehogSummary: Hedgehog拮抗剂
- A3145 Afatinib dimaleate中文名: 马来酸阿法替尼Target: EGFR|HER2Summary: EGFR抑制剂
- A8528 TAK-285Target: EGFR|HER2Summary: HER2/EGFR(HER1)抑制剂