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- A8366 ARRY-380Target: HER2Summary: 酪氨酸激酶HER2和P95-HER2抑制剂。
- B1299 1-NM-PP1Target: Cyclin-Dependent Kinases|Bcr-Abl|Src|Ca2 /calmodulin-dependent protein kinases (CaMKs)|c-FynSummary: Pp60c-src抑制剂
- B1079 BMS-303141Target: ATP Citrate LyasesSummary: 有效的ATP-柠檬酸裂合酶抑制剂
- A3145 Afatinib dimaleate中文名: 马来酸阿法替尼Target: EGFR|HER2Summary: EGFR抑制剂
- A8528 TAK-285Target: EGFR|HER2Summary: HER2/EGFR(HER1)抑制剂