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- A3237 Betulinic acid中文名: 白桦脂酸,桦木酸Target: Aminopeptidases|Topoisomerases|HIVSummary: 抗HIV和抗肿瘤化合物,五环三萜类化合物
- B1810 Penfluridol中文名: 五氟利多Target: Voltage-gated Calcium Channels (CaV)Summary: 多巴胺受体拮抗剂
- A3604 Mibefradil中文名: 米贝拉地尔,米贝地尔,咪拉地尔,咪贝地尔Target: Voltage-gated Calcium Channels (CaV)Summary: 钙通道阻滞剂
- B4745 (S)-10-Hydroxycamptothecin中文名: 羟喜树碱Target: TopoisomerasesSummary: 拓扑异构酶I抑制剂
- B1505 Epiandrosterone中文名: 表雄酮Target: Voltage-gated Calcium Channels (CaV)Summary: 类固醇激素,具有弱雄激素活性
- B1988 Nifedipine2 Citation中文名: 硝苯地平Target: Voltage-gated Calcium Channels (CaV)Summary: L-型钙通道阻断剂
- B1572 LatrepirdineTarget: Voltage-gated Calcium Channels (CaV)|NMDA receptor|adrenergic receptor|Histamine receptors|GluR|5-HT receptor|dopamine receptors|AMPA receptorSummary: 脑细胞死亡抑制剂
- B2278 Ibutilide Fumarate中文名: 富马酸伊布利特Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channelSummary: III类抗心律失常药物
- A8400 Clinafloxacin CI96 AM1091中文名: 克林沙星Target: TopoisomerasesSummary: 拓扑异构酶抑制剂
- A2601 Aclacinomycin ATarget: TopoisomerasesSummary: 拓扑异构酶I和II的双重抑制剂