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- A3020 (R)-Crizotinib2 Citation中文名: 克唑替尼Target: c-METSummary: ATP竞争性的C-MET/ALK抑制剂。
- A3433 Gefitinib hydrochloride中文名: 盐酸吉非替尼Target: EGFRSummary: EGFR有效的抑制剂
- B1309 GNE-617 hydrochlorideTarget: NamptSummary: NAMPT抑制剂
- A8620 AZD-34633 CitationTarget: ALK|Insulin-like growth factors (IGFs)Summary: ALK/IGF1R抑制剂