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- A4096 Belinostat (PXD101)2 Citation中文名: 贝利司他Target: Histone Deacetylases (HDACs)Summary: 羟肟酸型HDAC抑制剂
- A8182 3-Deazaneplanocin A (DZNep) hydrochloride1 Citation中文名: 3-去氮腺嘌呤A盐酸盐Target: EZH2Summary: SAHH和EZH2抑制剂
- B2127 Rifapentine中文名: 利福喷丁Target: RNA PolymerasesSummary: 治疗肺结核的抗生素药物.
- A3021 GDC-0449 (Vismodegib)1 Citation中文名: 维莫德吉Target: P-glycoprotein (P-gp)|HedgehogSummary: Hedgehog拮抗剂
- A3433 Gefitinib hydrochloride中文名: 盐酸吉非替尼Target: EGFRSummary: EGFR有效的抑制剂
- B1474 FT-207 (NSC 148958)中文名: 替加氟Summary: DNA/RNA合成抑制剂
- N2416 Licochalcone B中文名: 甘草查尔酮 B
- A2168 Dovitinib (TKI-258, CHIR-258)2 Citation中文名: 多韦替尼Target: FLT3|VEGFR|PDGFR|c-Kit|FGFRSummary: 多靶点RTK抑制剂
- A8219 Gefitinib (ZD1839)3 Citation中文名: 吉非替尼Target: EGFRSummary: EGFR抑制剂