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- A3927 VS-5584 (SB2343)Target: PI3K|mTORSummary: MTOR/P13K抑制剂
- B2219 EHop-0161 CitationTarget: RacSummary: Rac1/Rac3 GTPase抑制剂
- A8620 AZD-34633 CitationTarget: ALK|Insulin-like growth factors (IGFs)Summary: ALK/IGF1R抑制剂
- A5112 XL147Target: PI3KSummary: PI3K选择性、可逆的抑制剂
- A2681 TGX-221Target: PI3KSummary: PI3K抑制剂