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- B1317 ML-323Target: Deubiquitinating enzymes (DUBs)Summary: USP1-UAF1抑制剂
- A8212 PR-619Target: Deubiquitinating enzymes (DUBs)Summary: 去泛素化酶(DUBs)抑制剂
- A8623 TOK-001中文名: 加来特龙,伽来特隆Target: Androgen Receptors|Cytochrome P450 (CYP450)Summary: CYP17抑制剂和雄激素受体(AR)拮抗剂
- A8394 CHIR-124Target: FLT3|GSK-3|Chk|PDGFRSummary: Chk1抑制剂