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- N1336 Chrysin中文名: 柯因,5,7-二羟黄酮Target: Estrogen and Related Receptors|Hypoxia Inducible Factors (HIFs)Summary: 抗炎和抗肿瘤试剂
- B2143 Tacrolimus (FK506)2 Citation中文名: 他克莫司Target: Peptidylprolyl isomerasesSummary: 大环内酯类钙调神经磷酸酶抑制剂,免疫抑制剂。
- A3021 GDC-0449 (Vismodegib)1 Citation中文名: 维莫德吉Target: P-glycoprotein (P-gp)|HedgehogSummary: Hedgehog拮抗剂
- A3956 ZosuquidarTarget: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)Summary: MDR调节剂