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- A1971 Etoposide4 Citation中文名: 依托泊苷Target: TopoisomerasesSummary: 拓扑异构酶II(Topo II)抑制剂
- A4383 Tolcapone中文名: 托卡朋Target: Catechol O-Methyltransferase (COMT)Summary: COMT抑制剂
- A3136 A-740003Target: P2X ReceptorsSummary: P2X7受体拮抗剂
- A4330 Isotretinoin中文名: 罗可坦,异维A酸Target: RARsSummary: 多巴胺β-羟化酶激活剂
- B1013 GSK1324726ATarget: BromodomainsSummary: BET蛋白抑制剂
- A3284 Cathepsin S inhibitor1 CitationTarget: CathepsinsSummary: 抑制MHCII抗原呈递