MEK1/2 - Melanoma
MEK1/2, also known as MAPKK (mitogen-activated protein kinase kinase), is a kinase enzyme which phosphorylates MAPK (mitogen-activated protein kinase).
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- B1135 GDC-0623Target: MEKSummary: MEK1抑制剂
- B1621 TAK-733Target: MEKSummary: MEK变构位点抑制剂
- A8374 AZD8330Target: MEKSummary: MEK 1/2抑制剂
- A5573 Pimasertib (AS-703026)Target: MEKSummary: MEK1/2抑制剂
- A3887 Trametinib DMSO solvate1 CitationTarget: MEKSummary: 变构MEK1/MEK2 激酶抑制剂
- A3018 Trametinib (GSK1120212)7 Citation中文名: 曲美替尼Target: MEKSummary: MEK1和MEK2抑制剂
- A3004 Vemurafenib (PLX4032, RG7204)9 Citation中文名: 维罗非尼Target: RafSummary: BRAF激酶抑制剂