Roquinimex
mRNA synthesis
In vitro transcription of capped mRNA with modified nucleotides and Poly(A) tail
Tyramide Signal Amplification (TSA)
TSA (Tyramide Signal Amplification), used for signal amplification of ISH, IHC and IC etc.
Phos Binding Reagent Acrylamide
Separation of phosphorylated and non-phosphorylated proteins without phospho-specific antibody
Cell Counting Kit-8 (CCK-8)
A convenient and sensitive way for cell proliferation assay and cytotoxicity assay
SYBR Safe DNA Gel Stain
Safe and sensitive stain for visualization of DNA or RNA in agarose or acrylamide gels.
Inhibitor Cocktails
Protect the integrity of proteins from multiple proteases and phosphatases for different applications.
Roquinimex (Linomide; PNU212616; ABR212616)是免疫刺激剂,能增强NK细胞活性和巨噬细胞的细胞毒性,抑制血管生成和TNFα的分泌。TNFα对DSS处理的小鼠进行Roquinimex的预防性给药,可明显减少结肠炎、MDS和CH降低的临床症状。此外,在 roquinimex 治疗的动物中,与DSS对照小鼠相比,MPO活性显着降低了50%以上。值得注意的是,在DSS治疗的小鼠中治疗性给药roquinimex也显着抑制了 MDS、CH 还原和 MPO 活性[1]。
参考文献:
[1]. Liu Q, Wang Y, Wan MX, Zhang XW, Andersson G, Hedlund G, Thorlacius H. Roquinimex inhibits dextran sodium sulfate-induced murine colitis. Inflamm Res. 2003 Feb;52(2):64-8. doi: 10.1007/s000110300002. PMID: 12665123.
Storage | Store at -20°C |
M.Wt | 308.34 |
Cas No. | 84088-42-6 |
Formula | C18H16N2O3 |
Synonyms | Linomide;FCF89;ABR212616 |
Solubility | ≥30.8 mg/mL in DMSO |
Chemical Name | 4-hydroxy-N,1-dimethyl-2-oxo-N-phenyl-1,2-dihydroquinoline-3-carboxamide |
SDF | Download SDF |
Canonical SMILES | O=C(C1=C(O)C2=C(N(C)C1=O)C=CC=C2)N(C)C3=CC=CC=C3 |
运输条件 | 蓝冰运输或根据您的需求运输。 |
一般建议 | 不同厂家不同批次产品溶解度各有差异,仅做参考。若实验所需浓度过大至产品溶解极限,请添加助溶剂助溶或自行调整浓度。溶液形式一般不宜长期储存,请尽快用完。 |
质量控制和MSDS
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