NVP-BAG956
Catalog No.
A3672
PI3K和PDK1抑制剂
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NVP-BAG956(BAG 956) is a potent, ATP-competitive and selective dual PI3K and PDK1 inhibitor in vitro and in vivo,with IC50 values to be 56, 444, 34, 117 and 240 nM for PI3K p110 alpha, beta, delta and gamma and PDK1 kinases, respectively.
| Physical Appearance | Red solid |
| Storage | Store at -20°C |
| M.Wt | 427.5 |
| Cas No. | 853910-02-8 |
| Formula | C28H21N5 |
| Synonyms | BAG 956 |
| Solubility | Soluble in DMSO |
| Chemical Name | 2-methyl-2-(4-(2-methyl-8-(pyridin-3-ylethynyl)-1H-imidazo[4,5-c]quinolin-1-yl)phenyl)propanenitrile |
| SDF | Download SDF |
| Canonical SMILES | CC1=NC2=CN=C3C=CC(C#CC4=CN=CC=C4)=CC3=C2N1C5=CC=C(C(C)(C#N)C)C=C5 |
| 运输条件 | 蓝冰运输或根据您的需求运输。 |
| 一般建议 | 不同厂家不同批次产品溶解度各有差异，仅做参考。若实验所需浓度过大至产品溶解极限，请添加助溶剂助溶或自行调整浓度。溶液形式一般不宜长期储存，请尽快用完。 |
