PI3K
PI3K (phosphatidylinositol-4,5-bisphosphate 3-kinase) is a family of enzymes involved in cellular functions such as cell growth, proliferation, differentiation, motility, survival and intracellular trafficking, which in turn are involved in cancer.
- A8499 PF-04691502Target: Akt|PI3K|mTORSummary: PI3K/mTOR (FRAP)抑制剂
- A8488 NVP-BGT226Target: PI3K|mTORSummary: 新型的PI3K/mTOR选择性抑制剂
- A8354 A66Target: PI3KSummary: P110α抑制剂
- A8346 BYL-7191 Citation中文名: 阿培利司Target: PI3KSummary: 选择性的PI3Kα抑制剂
- A1720 Duvelisib (IPI-145, INK1197)中文名: 杜韦利西布Target: PI3KSummary: PI3K-δ/PI3K-γ 抑制剂
- A5634 SAR245409 (XL765)Summary: mTOR/PI3K抑制剂
- A5478 AZD6482Target: PI3KSummary: PI3Kβ的有效选择性抑制剂
- A5449 PIK-93Summary: PI3Kγ/PI4KIIIβ/PI3Kα抑制剂
- A5176 AS-605240Target: PI3KSummary: PI 3-Kγ选择性抑制剂
- A2065 IC-87114Summary: PI3Kδ抑制剂