PDE
PDE (phosphodiesterases) catalyze the hydrolysis of cGMP and/or cAMP. Stimulus such as light, neurotransmitter and hormone trigger PDE to regulate various biological response including vascular smooth muscle proliferation/contraction, hormone secretion and plate aggregation etc.
- A4343 Dyphylline中文名: 二羟丙茶碱Summary: Pan-PDE抑制剂
- A4340 Pimobendan中文名: 匹莫苯丹,匹莫苯Target: Phosphodiesterases (PDEs)Summary: PDE3抑制剂和Ca2+通道敏化剂
- A4337 Cilostazol中文名: 西洛他唑Summary: PDE3抑制剂
- A4334 Avanafil中文名: 阿伐那非Target: Phosphodiesterases (PDEs)Summary: PDE5抑制剂
- A4331 GSK256066Summary: PDE4的高效选择性抑制剂
- A4329 Cilomilast中文名: 西洛司特Target: Phosphodiesterases (PDEs)Summary: PDE4抑制剂
- A4328 Rolipram中文名: 咯利普兰Target: Phosphodiesterases (PDEs)Summary: PDE4抑制剂和抗炎剂
- A4327 Tadalafil中文名: 他达拉非Target: Phosphodiesterases (PDEs)Summary: PDE5抑制剂
- A4325 PF-2545920Target: Phosphodiesterases (PDEs)Summary: PDE10A的有效选择性抑制剂
- A4323 Vardenafil HCl Trihydrate中文名: 盐酸伐地那非三水合物Target: Phosphodiesterases (PDEs)Summary: PDE5抑制剂