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Androgen Receptor - Animal Experiments

AR (androgen receptor) is a member of steroid hormone receptor and ligand-activated transcription factor. It plays a crucial role in prostate cellular proliferation and male sexual differentiation.

10 件产品

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  1. ODM-201
    A8452 ODM-201
    中文名: 达洛鲁胺
    Target: Androgen Receptors
    Summary: 新一代雄激素受体抑制剂
      ≥19.95 mg/mL
      insoluble in H2O
  2. Estradiol valerate
    B1506 Estradiol valerate
    中文名: 戊酸雌二醇
    Target: Estrogen and Related Receptors
    Summary: 雌激素受体激动剂
      ≥15.45 mg/mL
      insoluble in H2O
  3. Epiandrosterone
    B1505 Epiandrosterone
    中文名: 表雄酮
    Target: Voltage-gated Calcium Channels (CaV)
    Summary: 类固醇激素,具有弱雄激素活性
      ≥28.27 mg/mL
      insoluble in H2O
  4. TOK-001
    A8623 TOK-001
    中文名: 加来特龙,伽来特隆
    Target: Androgen Receptors|Cytochrome P450 (CYP450)
    Summary: CYP17抑制剂和雄激素受体(AR)拮抗剂
      ≥12.4 mg/mL
      insoluble in H2O
  5. ARN-509
    A8364 ARN-509
     2 Citation
    中文名: 阿帕鲁胺
    Target: Androgen Receptor
    Summary: 雄激素受体抑制剂
      ≥23.85 mg/mL
      insoluble in H2O
  6. Andarine
    A2150 Andarine
    Target: Androgen Receptors
    Summary: 雄激素受体拮抗剂
      ≥21 mg/mL
      insoluble in H2O
  7. Bicalutamide
    A5065 Bicalutamide
     1 Citation
    中文名: 比卡鲁胺
    Target: Androgen Receptors
    Summary: 雄激素受体(Androgen receptor)拮抗剂
      ≥42.89 mg/mL
      insoluble in H2O
  8. ASC-J9
    A3190 ASC-J9
    中文名: 二甲基姜黄素
    Summary: AR降解的增强子,抗肿瘤剂
      ≥16.65 mg/mL
      insoluble in H2O
  9. TAK-700 (Orteronel)
    A4326 TAK-700 (Orteronel)
     2 Citation
    Target: human lyase
    Summary: 人17,20-裂解酶抑制剂
      ≥11.2 mg/mL
      insoluble in H2O
  10. MDV3100 (Enzalutamide)
    A3003 MDV3100 (Enzalutamide)
     12 Citation
    中文名: 恩杂鲁胺
    Target: Androgen Receptors
    Summary: 雄激素受体拮抗剂。
      ≥23.22 mg/mL
      insoluble in H2O

10 件产品

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