Androgen Receptor
AR (androgen receptor) is a member of steroid hormone receptor and ligand-activated transcription factor. It plays a crucial role in prostate cellular proliferation and male sexual differentiation.
- A1372 AZD3514Summary: 雄激素受体下调剂
- A2150 AndarineTarget: Androgen ReceptorsSummary: 雄激素受体拮抗剂
- A2961 MK-2866 (GTx-024)Summary: 雄激素受体调节剂
- A5065 Bicalutamide1 Citation中文名: 比卡鲁胺Target: Androgen ReceptorsSummary: 雄激素受体(Androgen receptor)拮抗剂
- A3780 RU 58841Summary: 雄激素受体拮抗剂
- A3190 ASC-J9中文名: 二甲基姜黄素Summary: AR降解的增强子,抗肿瘤剂
- A3108 17 alpha-propionateSummary: 雄激素拮抗剂
- A4326 TAK-700 (Orteronel)2 CitationTarget: human lyaseSummary: 人17,20-裂解酶抑制剂
- A3003 MDV3100 (Enzalutamide)12 Citation中文名: 恩杂鲁胺Target: Androgen ReceptorsSummary: 雄激素受体拮抗剂。