Androgen Receptor
AR (androgen receptor) is a member of steroid hormone receptor and ligand-activated transcription factor. It plays a crucial role in prostate cellular proliferation and male sexual differentiation.
- B7503 Cl-4AS-1Summary: 类固醇雄激素受体激动剂
- B7468 CITCO1 CitationTarget: constitutive androstane receptor (CAR)Summary: 组成型雄激素受体(CAR)激动剂
- B7536 PF 998425Summary: 非类固醇雄激素受体(AR)拮抗剂
- B1378 Spironolactone1 Citation中文名: 螺内酯Summary: 竞争性盐皮质激素(醛固酮)受体拮抗剂
- B1376 Flutamide中文名: 氟他胺Summary: 雄激素受体拮抗剂
- B1506 Estradiol valerate中文名: 戊酸雌二醇Target: Estrogen and Related ReceptorsSummary: 雌激素受体激动剂
- B1505 Epiandrosterone中文名: 表雄酮Target: Voltage-gated Calcium Channels (CaV)Summary: 类固醇激素,具有弱雄激素活性
- A8623 TOK-001中文名: 加来特龙,伽来特隆Target: Androgen Receptors|Cytochrome P450 (CYP450)Summary: CYP17抑制剂和雄激素受体(AR)拮抗剂
- A8404 Cyproterone Acetate中文名: 醋酸环丙氯地孕酮Summary: 雄激素受体拮抗剂
- A8364 ARN-5092 Citation中文名: 阿帕鲁胺Target: Androgen ReceptorSummary: 雄激素受体抑制剂