VEGFR
VEGFR are receptors for vascular endothelial growth factor and belong to receptor tyrosine kinases.
- A8418 Dovitinib Dilactic acidSummary: FLT3抑制剂
- A8370 Axitinib (AG 013736)1 Citation中文名: 阿西替尼Target: VEGFR|PDGFR|c-KitSummary: VEGFR1/ c-Kit抑制剂
- A8347 Pazopanib Hydrochloride中文名: 盐酸帕佐帕尼Summary: VEGFR/PDGFR/FGFR/c-Kit/ c-Fms抑制剂
- A8313 RAF265Target: Raf|VEGFRSummary: 多细胞激酶抑制剂
- A5760 KRN 633Summary: VEGFR的ATP竞争性抑制剂
- A5467 Ponatinib (AP24534)1 Citation中文名: 帕纳替尼Target: VEGFR|PDGFR|Bcr-Abl|FGFR|SrcSummary: pan-BCR-ABL抑制剂,多激酶抑制剂
- A5331 TSU-68 (SU6668,Orantinib)Summary: PDGFR/Flk-1/FGFR1的强效竞争性抑制剂
- A1778 Vatalanib (PTK787) 2HCl中文名: 瓦他拉尼二盐酸盐Target: VEGFRSummary: 酪氨酸激酶受体抑制剂
- A2633 Brivanib Alaninate (BMS-582664)中文名: 丙氨酸布立尼布Summary: VEGFR2的ATP竞争性抑制剂
- A2974 Foretinib (GSK1363089)1 CitationSummary: VEGF和HGF受体抑制剂