PI3K
PI3K (phosphatidylinositol-4,5-bisphosphate 3-kinase) is a family of enzymes involved in cellular functions such as cell growth, proliferation, differentiation, motility, survival and intracellular trafficking, which in turn are involved in cancer.
- A2080 PIK-75 HClSummary: PI3K亚型p110α抑制剂
- A2764 PIK-90Summary: 有效的PI3K选择性抑制剂
- A2754 TG100-115Target: PI3KSummary: PI3Kγ/PI3Kδ抑制剂
- A2552 Quercetin dihydrate中文名: 槲黄素,槲皮素二水化物Target: PI3K|PIM1 kinase|phospholipase A2Summary: PLA2和PI3K抑制剂
- A2681 TGX-221Target: PI3KSummary: PI3K抑制剂
- A5112 XL147Target: PI3KSummary: PI3K选择性、可逆的抑制剂
- A2067 PI-1031 CitationSummary: I类PI3K、mTOR和DNA-PK抑制剂
- A8250 LY 29400216 CitationTarget: PI3KSummary: PI3K抑制剂
- A8248 ZSTK474Summary: PI3K的强效抑制剂
- A8246 BEZ235 (NVP-BEZ235)2 Citation中文名: 达克利司Summary: ATP竞争性的PI3K/mTOR抑制剂