CYP3A/CYP450
CYP3A4 is an enzyme of cytochrome P450 superfamily found in human liver. It catalyzes the metabolism of endogenous and exogenous agents ( e.g. xenobiotics).
- B5724 Pentoxyresorufin中文名: 7-羟基吩噁嗪酮二戊醚Summary: 荧光细胞色素P450底物
- B5723 Methoxyresorufin中文名: 甲氧基试卤灵Summary: 细胞色素P450的荧光底物
- B7737 ABT中文名: 1-氨基苯并三唑Summary: 细胞色素P450抑制剂
- A3374 Dronedarone中文名: 决奈达隆Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channelSummary: CYP3A4和2D6抑制剂
- A4322 Clarithromycin中文名: 克拉霉素Target: Cytochrome P450 (CYP450)Summary: CYP3A抑制剂
- A4320 Voriconazole中文名: 伏立康唑Summary: CYP51抑制剂
- A4313 Cobicistat (GS-9350)中文名: 可比司他Target: Cytochrome P450 (CYP450)Summary: CYP3A的选择性抑制剂