EGFR
EGFR (epidermal growth factor receptor) is the cell-surface receptor of its specific ligands, including epidermal growth factor and TGFα (transforming growth factor α) and is a receptor tyrosine kinase.
- A5455 AEE788 (NVP-AEE788)Summary: EGFR/HER-2/VEGFR抑制剂
- A1845 Canertinib (CI-1033)中文名: 卡奈替尼Summary: HER家族酪氨酸激酶抑制剂
- A1393 WZ8040Target: EGFRSummary: EGFR T790M抑制剂
- A1835 Pelitinib (EKB-569)中文名: 培利替尼Summary: 有效的EGFR不可逆抑制剂
- A2412 CP-724714Target: VEGFR|PDGFR|Bcr-Abl|Src|EGFR|c-MET|Insulin Receptors|IRG-1RSummary: 有效的HER2选择性抑制剂
- A1389 WZ4002Summary: 突变型(L858R,T790M)EGFR抑制剂
- A8247 Afatinib (BIBW2992)1 Citation中文名: 阿法替尼Target: EGFRSummary: EGFR/ HER2抑制剂
- A8234 Erlotinib Hydrochloride2 Citation中文名: 盐酸厄洛替尼Summary: EGFR抑制剂
- A8219 Gefitinib (ZD1839)3 Citation中文名: 吉非替尼Target: EGFRSummary: EGFR抑制剂
- A8218 Lapatinib2 Citation中文名: 拉帕替尼Target: ErbBSummary: EGFR/HER2抑制剂