Androgen Receptor - Selective
AR (androgen receptor) is a member of steroid hormone receptor and ligand-activated transcription factor. It plays a crucial role in prostate cellular proliferation and male sexual differentiation.
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- B1505 Epiandrosterone中文名: 表雄酮Target: Voltage-gated Calcium Channels (CaV)Summary: 类固醇激素,具有弱雄激素活性
- A8623 TOK-001中文名: 加来特龙,伽来特隆Target: Androgen Receptors|Cytochrome P450 (CYP450)Summary: CYP17抑制剂和雄激素受体(AR)拮抗剂
- A8364 ARN-5092 Citation中文名: 阿帕鲁胺Target: Androgen ReceptorSummary: 雄激素受体抑制剂
- A2150 AndarineTarget: Androgen ReceptorsSummary: 雄激素受体拮抗剂
- A5065 Bicalutamide1 Citation中文名: 比卡鲁胺Target: Androgen ReceptorsSummary: 雄激素受体(Androgen receptor)拮抗剂
- A4326 TAK-700 (Orteronel)2 CitationTarget: human lyaseSummary: 人17,20-裂解酶抑制剂
- A3003 MDV3100 (Enzalutamide)12 Citation中文名: 恩杂鲁胺Target: Androgen ReceptorsSummary: 雄激素受体拮抗剂。